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OpenSourceMalaria
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Series4
Repository for Series 4 of the Open Source Malaria Consortium
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Next batch of compounds sent for testing April and June 2024
#79
qxsml
opened
5 months ago
19
Incorporation of data from two Davis et al papers
#78
mattodd
opened
1 year ago
2
Next batch of compounds sent for testing June 2021
#77
kym834
opened
1 year ago
0
Unexpected isomerization of oxetane-carboxylic acids
#76
mattodd
opened
2 years ago
1
My OSM PhD is complete!
#75
edwintse
opened
4 years ago
3
Which intermediates should we make? - OSM at Federation Uni
#74
david1597
opened
4 years ago
33
Next batch of compounds sent for biological testing August 2019 Sydney
#73
maratsydney
opened
5 years ago
2
July 2019 Compounds for Metabolic/Physchem Evaluation
#72
edwintse
opened
5 years ago
7
Next batch of compounds sent for biological testing Jul 2019
#71
edwintse
opened
5 years ago
8
Write-up of the Predictive Modelling Competition Results
#70
edwintse
closed
5 years ago
5
KinomeScan of Series 4 and telesubstitution compounds
#69
maratsydney
opened
5 years ago
3
Master list
#68
cdsouthan
closed
5 years ago
1
Remaining Data Needed for OHOH Compound(s)
#67
mattodd
opened
5 years ago
0
Poster that was presented at RACI 2018 organic conference
#66
maratsydney
closed
5 years ago
2
November 2018 Potency results
#65
mbhebhe
opened
5 years ago
10
CO-ADD assay
#64
MFernflower
closed
5 years ago
10
Compounds for hERG Evaluation Round 2
#63
edwintse
opened
5 years ago
6
Compounds sent for biological testing Nov 2018
#62
mbhebhe
closed
5 years ago
15
Compounds for biological testing Nov 2018
#61
maratsydney
closed
5 years ago
1
Exploration of 6-substituted compounds
#60
maratsydney
opened
5 years ago
20
Potency results on the repeated biotransformation
#59
david1597
opened
6 years ago
2
Possible enantioselective synthetic route to the OHOH compounds
#58
david1597
closed
6 years ago
2
DCNYS question
#57
MFernflower
closed
6 years ago
1
April 2018 Dundee Potency Results
#56
david1597
closed
4 years ago
5
Ring expanded analogues of the indole hit
#55
MFernflower
opened
6 years ago
4
Next batch of compounds sent for biological testing June 2018
#54
edwintse
opened
6 years ago
6
2018 SSP Compounds
#53
edwintse
opened
6 years ago
30
Lipophilic Efficiency
#52
david1597
opened
6 years ago
1
Series 4 Synthesis Update - June 2018
#51
david1597
closed
6 years ago
2
Exploration of benzylic amines
#50
david1597
opened
6 years ago
2
5-S-linked pyrazine side chains
#49
edwintse
closed
6 years ago
12
Revising/correcting our data on N/S linked pyrazine side chain compounds
#48
david1597
opened
6 years ago
2
5-N-linked pyrazine side chains
#47
david1597
opened
6 years ago
19
The Aussies - unexpected products from substitution down under
#46
david1597
opened
6 years ago
10
Cyclopropyloxy and other abnormal RHS para-ethers
#45
MFernflower
opened
6 years ago
0
Further exploration of benzylic alcohols (and a faster route to them)
#44
david1597
opened
6 years ago
12
Possible new linkers on the LHS at Griffith Uni: Carbamates and Ureas
#43
Plebellec
opened
6 years ago
19
May 2018 Compounds for Metabolic/Physchem Evaluation
#42
edwintse
opened
6 years ago
13
The side-products formed during The OHOH synthesis
#41
david1597
closed
6 years ago
3
Next Series 4 targets at Griffith Uni - comments and suggestions
#40
mcoster
closed
6 years ago
12
April 2018 Shipment for biological activity evaluation to Dundee
#39
maratsydney
opened
6 years ago
61
The Nemesis has been successfully synthesised
#38
edwintse
closed
6 years ago
3
April 2018 Compounds for hERG Evaulation
#37
edwintse
closed
6 years ago
15
Synthesis of "The OHOH" - a benzylic hydroxylation product
#36
david1597
opened
6 years ago
23
Liver stage results
#35
david1597
closed
3 years ago
5
Questions about LHS benzene ring halogenation
#34
MFernflower
closed
6 years ago
1
Identification of the compound made in the original bio-transformation experiment
#33
david1597
opened
6 years ago
24
Which compounds should we send for biofunctionalisation (batch III) April 2018?
#32
david1597
closed
6 years ago
11
New set of boronic acids based on new hit OSM-S-525 + some others
#31
maratsydney
opened
6 years ago
19
The Phenylalaninol ether has been successfully synthesised
#30
edwintse
closed
6 years ago
3
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